Cardarine GW 501516


Have you heard of Cardarine GW 501516? It is a research chemical that has recently received a lot of attention due to its potential benefits for improving endurance, stamina, and other health benefits.

But what exactly is Cardarine GW 501516, and how does it work? The information provided below provides an overview of Cardarine GW 50516.

It’s important to keep in mind that Cardarine GW 501516, along with other research compounds, is intended only for research purposes and not for human consumption. offers this product only for sale for research use and does not endorse or recommend it for any other purpose. If you are using this product for research, be sure to follow all handling instructions and safety precautions.

Cardarine GW 501516 Product Details

GW501516 ( or Cardarine ) is a research chemical that was developed in the 1990s to prevent and cure tumor formation in the colon, prostate, and breasts in humans. The purpose of developing Cardarine GW 501516 as a selective androgen receptor modulator (SARM) was to assist in the treatment of diseases like diabetes, obesity, and cardiovascular disease. It has also been discovered to have some potential fascinating effects on fat burning and endurance, which has increased its appeal to physical fitness activities. It process by attaching and activating the PPAR-delta protein, which then causes the body to undergo several metabolic changes. (R)(R) (R)

Here is the chemical composition of Cardarine GW 501516: (R)Product Name: Cardarine GW 501516 
Application: Scientific
CAS: 317318-70-0
Molar Mass: 453.49 g·mol−1
Chemical Formula: C21H18F3NO3S2
IUPAC Name: {4-[({4-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-thiazol-5-yl}methyl)sulfanyl]-2-methylphenoxy}acetic acid
Synonyms: GW-501; 516; GW1516; GSK-516, Cardarine
Storage:  Minimize open-air exposure, store in a cool dry place
Variants: Cardarine GW 501516 powder (1000mg) and Liquid (30ml/ 33mg per ml/ 1000mg) (30ml/ 67mg per ml/ 2000mg)

How Does Cardarine GW 501516 Work?

Cardarine GW 501516 functions by turning on a particular protein known as PPAR-delta. Nuclear receptor PPAR-delta alters the expression of specific genes, which affects the body’s physiology and metabolism. Cardarine can increase the potential expression of genes involved in the oxidation of fatty acids for energy when it binds to PPAR-delta. This implies that more fat can be utilized as a source of energy during physical activity, which can help increase energy levels and encourage weight loss. (R)(R)

By increasing the amount of oxygen delivered to muscles, Cardarine GW 501516 can potentially help improve endurance during exercise. Cardarine does this by activating the PPAR-delta protein, which stimulates the release of the hormone erythropoietin (EPO). During exercise, EPO stimulates the production of new red blood cells, which transport oxygen to muscles. If muscles have more oxygen, physical activity can be done for longer periods and perform better. (R)

Cardarine has also the potential for fat loss by increasing the activity of certain genes involved in fatty acid breakdown to eliminate excess fatty tissue and produce energy. This can lead to weight loss and increased energy levels while exercising and enhance recovery. While Cardarine has shown promising results in some clinical trials, more research is needed to fully understand it. (R)

What are the Potential Applications of Cardarine GW 501516?

Fat Metabolism

Cardarine has been shown to potentially improve the process of fat burning by increasing the body’s ability to use fatty acid metabolism decreasing the amount of carbohydrates or fat stored as adipose tissue. The body fat pushes skeletal muscle cells towards preferential lipid utilization and fat burning. Cardarine significantly increased the expression of genes involved in fatty acid oxidation while decreasing the expression of genes involved in fat storage in a clinical study on obese mice. The study concluded that Cardarine could be used to treat obesity and related metabolic disorders. (R) (R) (R)


Cardarine has been shown to potentially improve endurance by increasing red blood cell production, which improves oxygen delivery to the muscles during exercise. Cardarine increased endurance capacity in rats by 45% when compared to a control group in a clinical study. (R)

Cardiovascular Illness

Cardarine has been discovered to have potential cardiovascular disease benefits by improving lipid and glucose metabolism. Cardarine significantly reduced total cholesterol, triglycerides, and LDL cholesterol while increasing HDL cholesterol in a clinical study on mice with high cholesterol levels. The study concluded that Cardarine could be used to treat hyperlipidemia and other cardiovascular diseases. (R)


Cardarine has been shown to potentially improve glucose metabolism and decrease insulin resistance, which may have diabetes-related benefits. Cardarine improved glucose tolerance and insulin sensitivity while decreasing inflammation and oxidative stress in diabetic mice, according to a clinical study. The study concluded that Cardarine could be used to treat type 2 diabetes and other metabolic disorders. (R) (R)

Safety and Side Effects

  1. Potential Cancer Risk: Some animal studies have suggested that Cardarine may increase the potential risk of cancer, especially in the liver. It should be noted, however, that more research is needed to fully understand this potential risk. (R)
  2. Negative Impact on Cholesterol Levels: Cardarine hurts cholesterol levels, according to some studies. It can lower HDL (good) cholesterol levels while increasing LDL (bad) cholesterol levels. One may be more susceptible to heart disease as a result of this. (R)
  3. Liver Damage: Cardarine has occasionally been linked to liver damage or abnormalities in liver function. (R)
  4. Other Potential Side Effects: It also has mentioned experiencing fatigue, nausea, and headaches. Most of the time, these side effects are minor and go away on their own. (R)

In addition, the regulatory status of Cardarine remains unclear. The compound has not been approved for use by the US Food and Drug Administration (FDA) or other regulatory agencies, and its legal status varies from country to country. (R) (R)


Cardarine GW 501516’s future is currently unknown. There are still many unanswered questions regarding the drug’s safety and effectiveness in humans, even though preclinical and early-stage clinical studies have suggested potential benefits. 

But, as with many research substances, it’s always possible that more investigation will yield fresh insights and Cardarine’s potential uses. We might learn more about this substance’s effectiveness and safety as researchers continue to examine its mechanisms of action and potential applications.

The outcome of ongoing research, as well as legislative choices, will ultimately determine Cardarine’s future. Even though it is impossible to foresee exactly what will happen to Cardarine in the future, we can be sure that in the years to come, researchers and scientists will continue to examine its potential applications and safety profile. (R) (R)


What is Cardarine GW 501516?

A: Cardarine is a research compound that has been shown to have potential benefits in increasing endurance, burning fat, and improving metabolic health.

How does Cardarine work?

A: Cardarine works by activating the PPAR-delta pathway in the body, which has been linked to various metabolic and physiological effects, including increased endurance and fat burning in skeletal muscle tissue, and alleviates metabolic syndrome. The body fat pushes skeletal muscle cells towards preferential lipid utilization and fat burning.

Is Cardarine safe?

While Cardarine has shown potential benefits in research studies, there are also potential safety concerns and side effects associated with its use, such as an increased risk of cancer and a negative impact on cholesterol levels. It’s important to use Cardarine responsibly and under the guidance of a healthcare provider.

Will there be further research on Cardarine?

There may be further research on Cardarine in the future, particularly in terms of its potential benefits and safety concerns. However, any research will need to be carefully conducted and evaluated to ensure that it is conducted safely and ethically.

Is Cardarine legal?

The legal status of Cardarine varies depending on the country and jurisdiction in which it is being used. In some areas, Cardarine is considered a banned substance and its use is strictly prohibited. In other areas, it may be available for research purposes. It is important to check the legal status of Cardarine in your area before using it.

Can Cardarine be used for athletic performance enhancement?

Cardarine is not approved for use as a performance-enhancing drug, and its use in competitive sports is generally prohibited. Athletes who are subject to drug testing should be aware of the potential risks associated with Cardarine use and should avoid using it unless it is explicitly allowed by the relevant sports governing body.

Can Cardarine be used for medical purposes?

Cardarine is not currently approved for medical use by regulatory agencies such as the US FDA. However, there may be some potential therapeutic applications of Cardarine, particularly in the treatment of metabolic disorders such as obesity and type 2 diabetes. Any medical use of Cardarine would need to be carefully evaluated and approved by regulatory agencies.

Where to Buy Cardarine GW 501516?

When it comes to Nootropics and other research compounds is among the most reliable and novel companies available. We offer targeted solutions with lab-tested purity for your specific needs.


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